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N-(2-Chloro-4-hydroxyphenyl)-N'-cyclopropyl-urea CAS: 796848-79-8
N-(2-Chloro-4-hydroxyphenyl)-N'-cyclopropyl-urea yog ib qho tshuaj sib xyaw nrog cov mis molecular C10H11ClN2O2. Nws yog ib feem ntawm cov chav kawm ntawm urea derivatives hloov nrog ib pawg chloro-hydroxyphenyl thiab ib pawg cyclopropyl. Cov tshuaj no tau lees paub rau nws qhov nyuaj ntawm cov qauv thiab cov peev xwm siv hauv ntau yam kev tshawb fawb txog tshuaj lom neeg thiab kab mob.
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1,4-Dihydro-7-methoxy-4-oxo-6-quinolinecarboxylic acid methyl ester CAS: 205448-65-3
1,4-Dihydro-7-methoxy-4-oxo-6-quinolinecarboxylic acid methyl ester yog ib qho tshuaj lom neeg uas muaj cov mis molecular C12H11NO4. Nws yog ib feem ntawm cov tshuaj quinoline thiab nws yog ib pawg methyl ester uas txuas nrog lub nplhaib quinoline, nrog rau ib pawg methoxy substituent ntawm txoj haujlwm 7 thiab ib pawg keto ntawm txoj haujlwm 4.
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AZD-9291 mesylate CAS: 1421373-66-1
AZD-9291 mesylate yog ib qho tshuaj uas muaj cov mis molecular C28H33N7O4∙CH4O3S. Nws yog ib hom tshuaj uas ua rau cov tshuaj tyrosine kinase inhibitors tsis ua haujlwm thiab feem ntau yog siv rau kev kho mob qog nqaij hlav hauv lub ntsws uas tsis yog qog me me (NSCLC). Cov tshuaj no xaiv cov tshuaj uas tiv thaiv thiab tiv thaiv cov hlwb uas hloov pauv ntawm cov hlwb epidermal growth factor receptor (EGFR), uas feem ntau pom muaj nyob rau hauv cov qog NSCLC.
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5-Chloromethyl-2H-1,2,4-triazolin-3-ib CAS: 252742-72-6
5-Chloromethyl-2H-1,2,4-triazolin-3-one yog ib qho tshuaj lom neeg tseem ceeb uas siv tau ntau yam hauv kev kho mob thiab kev tshawb fawb txog kev ua liaj ua teb. Nws yog ib feem ntawm pawg triazolinone derivatives, uas muaj cov qauv molecular tshwj xeeb uas pab txhawb rau nws cov haujlwm biological thiab kev siv tshuaj kho mob.
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5-CHLOROTHIOPHENE-2-CARBONYL CHLORIDE CAS: 42518-98-9
5-Chlorothiophene-2-carbonyl chloride yog ib qho tshuaj lom neeg uas yog ib feem ntawm pawg thienylacyl chlorides. Nws yog tus cwj pwm los ntawm nws cov qauv molecular uas muaj lub nplhaib thiophene hloov nrog pawg chloro ntawm 5-txoj haujlwm thiab pawg carbonyl chloride ntawm 2-txoj haujlwm. Cov tshuaj no yog qhov txaus siab rau kev tsim cov organic vim nws cov tshuaj tiv thaiv ntau yam thiab cov ntawv thov hauv kev lag luam tshuaj thiab cov ntaub ntawv tshawb fawb.
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5,6-Dihydro-3-(4-morpholinyl)-1-(4-nitrophenyl)-2(1H)-pyridinone CAS:503615-03-0
5,6-Dihydro-3-(4-morpholinyl)-1-(4-nitrophenyl)-2(1H)-pyridinone yog ib hom tshuaj uas paub txog nws cov qauv molecular nyuaj thiab ntau yam kev siv hauv kev kho mob thiab kev tshawb fawb txog tshuaj. Cov tshuaj no yog ib hom pyridinones thiab nws muaj cov pab pawg ua haujlwm tshwj xeeb, uas muab cov yam ntxwv tshwj xeeb rau nws cov haujlwm hauv lub cev.
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4-Chloro-2-methylsulfanyl-pyrimidine-5-carboxylic acid ethyl ester CAS: 5909-24-0
4-Chloro-2-methylsulfanyl-pyrimidine-5-carboxylic acid ethyl ester yog ib qho tshuaj lom neeg uas paub txog nws lub luag haujlwm tseem ceeb hauv kev tshawb fawb txog tshuaj thiab kev tshawb fawb txog tshuaj. Ua ib feem ntawm cov pyrimidine derivatives, cov tshuaj no qhia txog cov qauv molecular tshwj xeeb uas tseem ceeb rau nws cov haujlwm biological thiab kev siv kho mob.
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3-CHLORO-4-METHOXYBENZYLAMINE HYDROCHLORIDE CAS: 41965-95-1
3-Chloro-4-Methoxybenzylamine Hydrochloride yog ib qho tshuaj lom neeg tseem ceeb uas paub dav dav rau nws cov kev siv hauv kev kho mob thiab kev tshawb fawb txog tshuaj. Cov tshuaj no poob rau hauv chav kawm ntawm cov amines aromatic thiab nws txawv los ntawm nws cov kev teeb tsa tshwj xeeb ntawm cov pab pawg ua haujlwm tseem ceeb rau nws cov haujlwm biological.
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3-Morpholino-1-(4-(2-oxopiperidin-1-yl)phenyl)-5,6-dihydropyridin-2(1H)-one CAS:545445-44-1
3-Morpholino-1-(4-(2-oxopiperidin-1-yl)phenyl)-5,6-dihydropyridin-2(1H)-one yog ib hom tshuaj uas paub zoo txog nws cov qauv molecular nyuaj thiab ntau yam kev siv hauv kev kho mob thiab kev tsim tshuaj. Cov tshuaj no yog ib hom dihydropyridinones thiab nws muaj cov pab pawg ua haujlwm sib txawv, uas muab cov yam ntxwv tshwj xeeb rau nws cov haujlwm hauv lub cev.
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L(-)-Thiazolidine-4-carboxylic acid CAS:34592-47-7
L(-)-Thiazolidine-4-carboxylic acid yog ib qho tshuaj lom neeg tseem ceeb uas paub txog nws cov kev siv ntau yam hauv kev kho mob thiab kev tshawb fawb txog tshuaj. Ua ib feem ntawm cov thiazolidine derivatives, cov tshuaj no muaj cov qauv molecular sib txawv rau nws cov haujlwm biological thiab lub peev xwm kho mob.
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Nintedanib CAS: 656247-17-5
Nintedanib yog ib qho tshuaj me me uas muaj zog tyrosine kinase inhibitor (TKI) nrog rau kev kho mob tseem ceeb hauv oncology thiab fibrotic kab mob. Nws ua rau nws cov teebmeem pharmacological los ntawm kev tsom mus rau ntau tus receptor tyrosine kinases uas koom nrog angiogenesis, fibrogenesis, thiab kev tswj kev loj hlob ntawm qog.
