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5-Bromo-2-chloro-4-(cyclopentylamino) pyrimidine CAS: 733039-20-8
5-Bromo-2-chloro-4-(cyclopentylamino) pyrimidine yog ib yam tshuaj uas tau tshawb nrhiav hauv kev tshawb fawb txog tshuaj. Nws muaj cov qauv pyrimidine nrog bromo thiab chloro hloov pauv, tej zaum yuav muaj txiaj ntsig zoo rau kev siv kho mob, tsom mus rau cov txheej txheem kab mob lossis cov kab mob hauv kev tshawb nrhiav tshuaj.
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4-[6-[[6-(1-Butoxyvinyl)-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino]pyridin-3-yl]piperazine-1-carboxylic acid tert-butyl ester CAS:866084-31-3
4-[6-[[6-(1-Butoxyvinyl)-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino]pyridin-3-yl]piperazine-1-carboxylic acid tert-butyl ester yog ib qho tshuaj lom neeg uas muaj lub hauv paus piperazine nrog cov pab pawg ua haujlwm suav nrog pyridine, pyrimidine, thiab tert-butyl ester. Nws cov qauv txhawb nqa cov ntawv thov hauv kev kho mob thiab kev tsim tshuaj vim nws cov tshuaj pharmacophores sib txawv.
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Bortezomib CAS: 179324-69-7
Bortezomib yog ib qho tshuaj siv los kho ntau yam mob myeloma thiab mantle cell lymphoma. Nws yog ib feem ntawm cov tshuaj proteasome inhibitors, uas tsom mus rau cov enzymes proteolytic hauv cov hlwb kom cuam tshuam lawv txoj haujlwm thiab ua rau apoptosis (programmed cell death). Lub tshuab no ua rau nws ua haujlwm zoo rau qee yam mob qog noj ntshav uas tsis tswj tau kev loj hlob ntawm cov hlwb.
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Methyl 2-bromomethyl-3-nitrobenzoate CAS: 98475-07-1
Methyl 2-bromomethyl-3-nitrobenzoate yog ib qho tshuaj lom neeg uas muaj ib pawg nitro ntawm 3-txoj hauj lwm thiab ib pawg bromomethyl ntawm 2-txoj hauj lwm ntawm ib qho benzoate backbone. Nws yog siv rau hauv kev tsim cov organic ua ib qho versatile intermediate, ua rau kev tsim cov molecules nyuaj nrog cov pab pawg ua haujlwm tshwj xeeb.
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Pemetrexed disodium INT-5 CAS: 165049-28-5
Pemetrexed disodium INT-5 yog ib hom tshuaj kho mob qog nqaij hlav uas raug muab faib ua cov tshuaj tua kab mob chemotherapy. Nws feem ntau yog siv rau kev kho mob ntau yam mob qog nqaij hlav, suav nrog mesothelioma, mob qog nqaij hlav ntsws non-small cell, thiab mob qog nqaij hlav metastatic tshwj xeeb.
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Pemetrexed disodium INT-4 CAS: 137281-39-1
Pemetrexed disodium INT-4 yog ib yam tshuaj tua kab mob chemotherapy uas siv rau hauv kev kho mob qog nqaij hlav. Nws siv rau kev kho mob ntau yam mob qog nqaij hlav, suav nrog mesothelioma, mob qog nqaij hlav ntsws non-small cell, thiab mob qog nqaij hlav metastatic tshwj xeeb.
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Pemetrexed disodium INT-3 CAS: 155405-80-4
Pemetrexed disodium INT-3 yog ib yam tshuaj tua kab mob chemotherapy uas siv rau hauv kev kho mob qog nqaij hlav. Nws siv rau kev kho mob ntau yam mob qog nqaij hlav, suav nrog mesothelioma, mob qog nqaij hlav ntsws non-small cell, thiab mob qog nqaij hlav metastatic tshwj xeeb.
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Terbinafine puag CAS: 91161-71-6
Terbinafine yog ib yam khoom xyaw tshuaj uas siv los kho cov kab mob fungal. Nws yog ib hom allylamine uas yog cov tshuaj tua kab mob fungal thiab paub txog nws cov txiaj ntsig zoo tiv thaiv dermatophytes, yeasts, thiab pwm.
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2-Chloro-4,6-dimethoxy-1,3,5-triazine CAS: 3140-73-6
2-Chloro-4,6-dimethoxy-1,3,5-triazine yog ib qho tshuaj lom neeg siv los ua ib qho khoom siv ntau yam hauv kev tsim cov organic thiab cov txheej txheem hloov kho tshuaj. Nws muaj cov pab pawg ua haujlwm chloro thiab methoxy txuas rau lub nplhaib triazine, ua rau nws siv tau rau ntau yam tshuaj lom neeg thiab cov qauv sib xyaw.
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2-Amino-4,5-bis(2-methoxyethoxy)benzonitrile CAS: 950596-58-4
2-Amino-4,5-bis(2-methoxyethoxy)benzonitrile yog ib qho tshuaj siv hauv kev tshawb fawb txog tshuaj, uas muaj cov qauv benzonitrile nrog cov amino thiab methoxyethoxy hloov chaw, uas tseem ceeb rau kev siv tshuaj kho mob tshwj xeeb.
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(1R)-(S)-pinanediol-1-Ammonium Trifluoroacetate-3-methlbutane-1-boronate CAS: 179324-87-9
(1R)-(S)-Pinanediol-1-Ammonium Trifluoroacetate-3-Methylbutane-1-Boronate yog ib qho tshuaj lom neeg uas muaj cov qauv nyuaj uas muaj pinanediol backbone, ib pawg ammonium trifluoroacetate, thiab ib qho boronate ester functionality. Nws yog siv rau hauv cov organic synthesis ua ib lub tsev chiral, ua rau muaj kev tsim cov tshuaj stereospecific thiab cov tshuaj intermediates.
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Diethyl L-glutamate hydrochloride CAS: 1118-89-4
Diethyl L-glutamate hydrochloride yog ib hom tshuaj siv feem ntau ua cov khoom siv nruab nrab hauv kev tshawb fawb txog tshuaj thiab kev tsim cov organic. Nws yog los ntawm L-glutamic acid thiab ua haujlwm ua tus thawj coj hauv kev tsim ntau yam tshuaj thiab cov tshuaj lom neeg.
